Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50045488
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064629(CHEMBL3403737)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064626(CHEMBL3403734)
Affinity DataKi:  334nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064637(CHEMBL3403727)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064636(CHEMBL3403726)
Affinity DataKi:  2.16E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064626(CHEMBL3403734)
Affinity DataKi:  2.38E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064631(CHEMBL3403739)
Affinity DataKi:  2.73E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064626(CHEMBL3403734)
Affinity DataKi:  3.44E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064630(CHEMBL3403738)
Affinity DataKi:  3.87E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064633(CHEMBL3403741)
Affinity DataKi:  3.91E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064620(CHEMBL3403728)
Affinity DataKi:  4.09E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064634(CHEMBL3403724)
Affinity DataKi:  4.12E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064621(CHEMBL3403729)
Affinity DataKi:  4.71E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064630(CHEMBL3403738)
Affinity DataKi:  5.67E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064634(CHEMBL3403724)
Affinity DataKi:  6.45E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064625(CHEMBL3403733)
Affinity DataKi:  7.13E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064620(CHEMBL3403728)
Affinity DataKi:  7.75E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064635(CHEMBL3403725)
Affinity DataKi:  8.22E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064628(CHEMBL3403736)
Affinity DataKi:  9.56E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064631(CHEMBL3403739)
Affinity DataKi:  9.66E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064637(CHEMBL3403727)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064629(CHEMBL3403737)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064627(CHEMBL3403735)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064624(CHEMBL3403732)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064627(CHEMBL3403735)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064637(CHEMBL3403727)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064627(CHEMBL3403735)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064631(CHEMBL3403739)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064621(CHEMBL3403729)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064633(CHEMBL3403741)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064625(CHEMBL3403733)
Affinity DataKi:  2.23E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064621(CHEMBL3403729)
Affinity DataKi:  2.35E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064633(CHEMBL3403741)
Affinity DataKi:  2.66E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064620(CHEMBL3403728)
Affinity DataKi:  2.84E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064628(CHEMBL3403736)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064635(CHEMBL3403725)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064636(CHEMBL3403726)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064632(CHEMBL3403740)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064632(CHEMBL3403740)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064622(CHEMBL3403730)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064636(CHEMBL3403726)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064635(CHEMBL3403725)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064632(CHEMBL3403740)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064630(CHEMBL3403738)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064629(CHEMBL3403737)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064628(CHEMBL3403736)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064623(CHEMBL3403731)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064623(CHEMBL3403731)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064625(CHEMBL3403733)
Affinity DataKi:  3.24E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064624(CHEMBL3403732)
Affinity DataKi:  3.40E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
B. V. Patel Pharmaceutical Education And Research Development (Perd) Centre

Curated by ChEMBL
LigandPNGBDBM50064623(CHEMBL3403731)
Affinity DataKi:  3.56E+4nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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