Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50046315
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105335BDBM50105335(CHEMBL3597247)
Affinity DataIC50: 280nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105353BDBM50105353(CHEMBL3597266)
Affinity DataIC50: 290nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105355BDBM50105355(CHEMBL3597268)
Affinity DataIC50: 410nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105333BDBM50105333(CHEMBL3597245)
Affinity DataIC50: 410nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105350BDBM50105350(CHEMBL3597264)
Affinity DataIC50: 510nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105354BDBM50105354(CHEMBL3597267)
Affinity DataIC50: 1.12E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105348BDBM50105348(CHEMBL3597262)
Affinity DataIC50: 1.44E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105349BDBM50105349(CHEMBL3597263)
Affinity DataIC50: 1.77E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50230993BDBM50230993(CHEMBL256147 | 2-Amino-5-(N'-methyl-guanidino)-pen...)
Affinity DataIC50: 2.30E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105344BDBM50105344(CHEMBL3597258)
Affinity DataIC50: 2.55E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105346BDBM50105346(CHEMBL3597260)
Affinity DataIC50: 2.57E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105351BDBM50105351(CHEMBL3597265)
Affinity DataIC50: 2.90E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105341BDBM50105341(CHEMBL3597254)
Affinity DataIC50: 3.43E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105334BDBM50105334(CHEMBL3597246)
Affinity DataIC50: 4.22E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105332BDBM50105332(CHEMBL3597244)
Affinity DataIC50: 4.43E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105345BDBM50105345(CHEMBL3597259)
Affinity DataIC50: 4.50E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105339BDBM50105339(CHEMBL3597252)
Affinity DataIC50: 4.51E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105342BDBM50105342(CHEMBL3597256)
Affinity DataIC50: 4.51E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105347BDBM50105347(CHEMBL3597261)
Affinity DataIC50: 4.54E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105331BDBM50105331(CHEMBL3597241)
Affinity DataIC50: 4.62E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105340BDBM50105340(CHEMBL3597253)
Affinity DataIC50: 4.66E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105343BDBM50105343(CHEMBL3597257)
Affinity DataIC50: 4.86E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Mouse)
Beni-Suef University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105337BDBM50105337(CHEMBL3597251)
Affinity DataIC50: 4.98E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed