Compile Data Set for Download or QSAR
maximum 50k data
Found 70 Enz. Inhib. hit(s) with all data for entry = 50045829
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084125(CHEMBL3425935)
Affinity DataIC50:  8nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084143(CHEMBL3425937)
Affinity DataIC50:  16nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084144(CHEMBL3425938)
Affinity DataIC50:  16nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084042(CHEMBL3425943)
Affinity DataIC50:  16nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084147(CHEMBL3425941)
Affinity DataIC50:  32nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084124(CHEMBL3425934)
Affinity DataIC50:  32nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084126(CHEMBL3425936)
Affinity DataIC50:  64nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084146(CHEMBL3425940)
Affinity DataIC50:  64nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084148(CHEMBL3425942)
Affinity DataIC50:  64nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084145(CHEMBL3425939)
Affinity DataIC50:  64nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084056(CHEMBL3425810)
Affinity DataIC50:  2.60E+3nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084055(CHEMBL3425808)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084049(CHEMBL3425806)
Affinity DataIC50:  1.17E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084110(CHEMBL3425822)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084043(CHEMBL3425798)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084045(CHEMBL3425800)
Affinity DataIC50:  2.77E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084122(CHEMBL3425931)
Affinity DataIC50:  2.82E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084052(CHEMBL3425807)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084049(CHEMBL3425806)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084114(CHEMBL3425825)
Affinity DataIC50:  3.04E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084048(CHEMBL3425805)
Affinity DataIC50:  3.05E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084120(CHEMBL3425929)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084115(CHEMBL3425826)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084123(CHEMBL3425932)
Affinity DataIC50:  3.36E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084119(CHEMBL3425927)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084116(CHEMBL3425827)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084121(CHEMBL3425930)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084046(CHEMBL3425801)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084047(CHEMBL3425802)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084118(CHEMBL3425926)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084057(CHEMBL3425811)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084099(CHEMBL3425812)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084100(CHEMBL3425813)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084102(CHEMBL3425814)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084104(CHEMBL3425816)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084105(CHEMBL3425817)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084107(CHEMBL3425818)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084108(CHEMBL3425819)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084109(CHEMBL3425820)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084111(CHEMBL3425823)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084112(CHEMBL3425514)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084113(CHEMBL3425824)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084116(CHEMBL3425827)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084117(CHEMBL3425924)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084118(CHEMBL3425926)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084119(CHEMBL3425927)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084117(CHEMBL3425924)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084121(CHEMBL3425930)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells measured over 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50068001(CHEMBL3400817)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50084044(CHEMBL3425799)
Affinity DataIC50: >6.00E+4nMAssay Description:Displacement of MK499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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