Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50046094
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094666(CHEMBL3589344)
Affinity DataKi:  42nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094667(CHEMBL3589343)
Affinity DataKi:  42nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50080827(CHEMBL333465 | (2R,6S)-1-Methyl-2,6-diphenethyl-pi...)
Affinity DataKi:  45nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094668(CHEMBL3589342)
Affinity DataKi:  57nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094667(CHEMBL3589343)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094706(CHEMBL3589345)
Affinity DataKi:  240nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094668(CHEMBL3589342)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094706(CHEMBL3589345)
Affinity DataKi:  627nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50094666(CHEMBL3589344)
Affinity DataKi:  647nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50080827(CHEMBL333465 | (2R,6S)-1-Methyl-2,6-diphenethyl-pi...)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50359499(METHAMPHETAMINE | (S)Methamphetamine)
Affinity DataKi:  2.46E+3nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50359499(METHAMPHETAMINE | (S)Methamphetamine)
Affinity DataKi:  8.01E+4nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2016
Entry Details Article
PubMed