Found 94 Enz. Inhib. hit(s) with all data for entry = 50046053 
Affinity DataKi: 0.5nMAssay Description:Displacement of (S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-((3H)-1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2 rec...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of (S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-((3H)-1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2 rec...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 137nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using paclitaxel as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 216nMAssay Description:Displacement of [3H]EMPA from human OX2 receptor expressed in human PFSK-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:Displacement of (S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-((3H)-1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2 rec...More data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Binding affinity to human OX1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 294nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 346nMAssay Description:Binding affinity to human OX1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 421nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 471nMAssay Description:Binding affinity to human OX1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 557nMAssay Description:Binding affinity to human OX1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 623nMAssay Description:Binding affinity to human OX1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 687nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 746nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 765nMAssay Description:Binding affinity to human OX1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 768nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 875nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
