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Found 18 Enz. Inhib. hit(s) with all data for entry = 50046348
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107317(CHEMBL3601177)
Affinity DataIC50:  7.30E+5nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107317(CHEMBL3601177)
Affinity DataIC50:  7.30E+5nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107321(CHEMBL3601173)
Affinity DataIC50:  8.80E+5nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107321(CHEMBL3601173)
Affinity DataIC50:  8.80E+5nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107320(CHEMBL3601174)
Affinity DataIC50:  9.10E+5nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107320(CHEMBL3601174)
Affinity DataIC50:  9.10E+5nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107319(CHEMBL3601175)
Affinity DataIC50:  9.70E+5nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107319(CHEMBL3601175)
Affinity DataIC50:  9.70E+5nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM22760(2-hydroxy-1,2-bis(4-methoxyphenyl)ethan-1-one | Be...)
Affinity DataIC50:  1.17E+6nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM22760(2-hydroxy-1,2-bis(4-methoxyphenyl)ethan-1-one | Be...)
Affinity DataIC50:  1.17E+6nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107318(CHEMBL3601176)
Affinity DataIC50:  1.29E+6nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107318(CHEMBL3601176)
Affinity DataIC50:  1.29E+6nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM22728(2-hydroxy-1,2-diphenylethan-1-one | Benzoin | CHEM...)
Affinity DataIC50:  2.12E+6nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM22728(2-hydroxy-1,2-diphenylethan-1-one | Benzoin | CHEM...)
Affinity DataIC50:  2.12E+6nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107322(CHEMBL3601172)
Affinity DataIC50:  2.66E+6nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107322(CHEMBL3601172)
Affinity DataIC50:  2.66E+6nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107316(CHEMBL3601178)
Affinity DataIC50:  2.82E+6nMAssay Description:Inhibition of PI3Kalpha in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Al-Zaytoonah University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50107316(CHEMBL3601178)
Affinity DataIC50:  2.82E+6nMAssay Description:Inhibition of PI3Kalpha H1047R mutant in human HCT116 cells assessed as cell growth inhibition after 24 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed