Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50046120
LigandChemical structure of BindingDB Monomer ID 50095475BDBM50095475(CHEMBL3590479)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095474BDBM50095474(CHEMBL3590478 | US10329294, Example 2)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50095470BDBM50095470(CHEMBL3590474 | US10155765, Example 9)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095532BDBM50095532(CHEMBL3590515 | US10329294, Example 173)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095534BDBM50095534(CHEMBL3590516 | US10329294, Example 252)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095473BDBM50095473(CHEMBL3590477 | US10329294, Example 282)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095531BDBM50095531(CHEMBL3590493 | US10329294, Example 60)
Affinity DataIC50: 1nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095505BDBM50095505(CHEMBL3590488 | US10329294, Example 88)
Affinity DataIC50: 1nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095465BDBM50095465(CHEMBL3590438 | US10155765, Example 28)
Affinity DataIC50: 2nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095476BDBM50095476(CHEMBL3590480 | US10329294, Example 297)
Affinity DataIC50: 2nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095514BDBM50095514(CHEMBL3590491 | US10329294, Example 205)
Affinity DataIC50: 3nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095517BDBM50095517(CHEMBL3590492)
Affinity DataIC50: 3nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095482BDBM50095482(CHEMBL3590486 | US10329294, Example 85)
Affinity DataIC50: 4nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095472BDBM50095472(CHEMBL3590476 | US10329294, Example 280)
Affinity DataIC50: 6nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095535BDBM50095535(CHEMBL3590517 | US10329294, Example 177)
Affinity DataIC50: 6nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095477BDBM50095477(CHEMBL3590481 | US10329294, Example 281)
Affinity DataIC50: 6nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095468BDBM50095468(CHEMBL3590473 | US10155765, Example 7)
Affinity DataIC50: 8nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095501BDBM50095501(CHEMBL3590487)
Affinity DataIC50: 10nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095509BDBM50095509(CHEMBL3590490 | US10329294, Example 97)
Affinity DataIC50: 13nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095471BDBM50095471(CHEMBL3590475 | US10329294, Example 279)
Affinity DataIC50: 14nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095467BDBM50095467(CHEMBL3590472)
Affinity DataIC50: 20nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095481BDBM50095481(CHEMBL3590485 | US10329294, Example 37)
Affinity DataIC50: 21nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095506BDBM50095506(CHEMBL3590489 | US10329294, Example 4)
Affinity DataIC50: 23nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095478BDBM50095478(CHEMBL3590482 | US10329294, Example 284)
Affinity DataIC50: 62nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095466BDBM50095466(CHEMBL3590471 | US10155765, Example 12)
Affinity DataIC50: 95nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095462BDBM50095462(CHEMBL3590435 | US10155765, Example 42)
Affinity DataIC50: 110nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095463BDBM50095463(CHEMBL3590436 | US9649308, Example 40)
Affinity DataIC50: 150nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095479BDBM50095479(CHEMBL3590483 | US10329294, Example 287)
Affinity DataIC50: 160nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095480BDBM50095480(CHEMBL3590484 | US10329294, Example 5)
Affinity DataIC50: 480nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50095464BDBM50095464(CHEMBL3590437 | US9649308, Example 39)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human IRAK4 assessed as phosphorylation of fluorescent peptide substrate after 30 mins by fluorescent polarization readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed