Affinity DataIC50: 13nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 158nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 176nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 726nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 2.88E+3nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMpH: 7.4Assay Description:hP2X7-expressing HEK 293 cells were re-suspended at 2.5 × 10^6 cells/mL in assay buffer composed of 10 mM HEPES, 5 mM N-methyl-D-glutamine, 5.6 mM KC...More data for this Ligand-Target Pair