Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50046361
TargetEndothelin-1 receptor(RAT)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50108104(CHEMBL3601500)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at endothelin A receptor in rat A7r5 cells assessed as inhibition of ET-1-induced increase in cytosolic free Ca2+ level treated 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Kansas State University

Curated by ChEMBL
LigandPNGBDBM50108104(CHEMBL3601500)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at endothelin A receptor in Wistar rat thoracic aorta strips assessed as inhibition of ET1-induced vasoconstriction preincubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed