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Found 13 Enz. Inhib. hit(s) with all data for entry = 50046846
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134204(CHEMBL3740772)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135099(CHEMBL3739636)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135098(CHEMBL3741585)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134208(CHEMBL3742039)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134205(CHEMBL3741102)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135104(CHEMBL3741981)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134206(CHEMBL3742032)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135101(CHEMBL3739701)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of UT-B in rat whole blood after 15 mins by RBC lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134207(CHEMBL3741384)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134203(CHEMBL2442435)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134202(CHEMBL424175)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135106(CHEMBL3739646)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of UT-B in rat whole blood after 15 mins by RBC lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135103(CHEMBL3741231)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed