Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50046524
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117151BDBM50117151(CHEMBL3613351)
Affinity DataIC50: 2nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117187BDBM50117187(CHEMBL3613341)
Affinity DataIC50: 5nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117149BDBM50117149(CHEMBL3613349)
Affinity DataIC50: 5nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117150BDBM50117150(CHEMBL3613355)
Affinity DataIC50: 5nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117149BDBM50117149(CHEMBL3613349)
Affinity DataIC50: 5nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117189BDBM50117189(CHEMBL3613340)
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117184BDBM50117184(CHEMBL3613347)
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117152BDBM50117152(CHEMBL3613350)
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117189BDBM50117189(CHEMBL3613340)
Affinity DataIC50: 12nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117153BDBM50117153(CHEMBL3613348)
Affinity DataIC50: 19nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117190BDBM50117190(CHEMBL3613339)
Affinity DataIC50: 22nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117152BDBM50117152(CHEMBL3613350)
Affinity DataIC50: 25nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117151BDBM50117151(CHEMBL3613351)
Affinity DataIC50: 32nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117190BDBM50117190(CHEMBL3613339)
Affinity DataIC50: 34nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117184BDBM50117184(CHEMBL3613347)
Affinity DataIC50: 44nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117153BDBM50117153(CHEMBL3613348)
Affinity DataIC50: 48nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117185BDBM50117185(CHEMBL3613344)
Affinity DataIC50: 69nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117187BDBM50117187(CHEMBL3613341)
Affinity DataIC50: 89nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117150BDBM50117150(CHEMBL3613355)
Affinity DataIC50: 105nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117185BDBM50117185(CHEMBL3613344)
Affinity DataIC50: 159nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117192BDBM50117192(CHEMBL3613357)
Affinity DataIC50: 170nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117146BDBM50117146(CHEMBL3613336)
Affinity DataIC50: 201nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117193BDBM50117193(CHEMBL3613356)
Affinity DataIC50: 280nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117194BDBM50117194(CHEMBL3613354)
Affinity DataIC50: 300nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117146BDBM50117146(CHEMBL3613336)
Affinity DataIC50: 491nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117200BDBM50117200(CHEMBL3613343)
Affinity DataIC50: 500nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117196BDBM50117196(CHEMBL3613352)
Affinity DataIC50: 500nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117195BDBM50117195(CHEMBL3613353)
Affinity DataIC50: 500nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117148BDBM50117148(CHEMBL3613334)
Affinity DataIC50: 539nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117148BDBM50117148(CHEMBL3613334)
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117186BDBM50117186(CHEMBL3613342)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117197BDBM50117197(CHEMBL3613346)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117199BDBM50117199(CHEMBL3613345)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117186BDBM50117186(CHEMBL3613342)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117145BDBM50117145(CHEMBL3613337)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117191BDBM50117191(CHEMBL3613338)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117147BDBM50117147(CHEMBL3613335)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117145BDBM50117145(CHEMBL3613337)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Mouse)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117147BDBM50117147(CHEMBL3613335)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse DGAT1 incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid scintillation counting and lumino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117191BDBM50117191(CHEMBL3613338)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human DGAT1 expressed in human Hep3B cells incubated for 60 mins using didecanoyl glycerol and [14C]decanoyl-CoA substrate by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 2(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50117149BDBM50117149(CHEMBL3613349)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human DGAT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed