Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50046547
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118105(CHEMBL3613443)
Affinity DataKi:  436nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118112(CHEMBL3613444)
Affinity DataKi:  777nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118110(CHEMBL3613449)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118111(CHEMBL3613442)
Affinity DataKi:  1.73E+3nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118109(CHEMBL3613448)
Affinity DataKi:  4.24E+3nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118107(CHEMBL3613446)
Affinity DataKi:  6.25E+3nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118106(CHEMBL3613445)
Affinity DataKi:  7.05E+3nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  8.82E+3nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50118108(CHEMBL3613447)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-astemizole from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed