Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50046717
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127666(CHEMBL3628839)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at S1P3 receptor (unknown origin) expressed in RBL membranes assessed as GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50127666(CHEMBL3628839)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at S1P1 receptor (unknown origin) expressed in CHO-K1 cells assessed as beta-arrestin recruitment after 60 mins by chemiluminescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed