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Found 16 Enz. Inhib. hit(s) with all data for entry = 50006378
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499318(CHEMBL3735996)
Affinity DataKi:  200nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499316(CHEMBL3734953)
Affinity DataKi:  700nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  920nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499316(CHEMBL3734953)
Affinity DataKi:  1.50E+3nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499318(CHEMBL3735996)
Affinity DataKi:  1.80E+3nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499315(CHEMBL3735566)
Affinity DataKi:  5.00E+3nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499317(CHEMBL3735043)
Affinity DataKi:  6.09E+3nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499315(CHEMBL3735566)
Affinity DataKi:  6.70E+3nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499313(CHEMBL3735387)
Affinity DataKi:  1.00E+4nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499312(CHEMBL3735271)
Affinity DataKi:  1.70E+4nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499314(CHEMBL3734842)
Affinity DataKi: >2.20E+4nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  3.60E+4nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499314(CHEMBL3734842)
Affinity DataKi: >6.00E+4nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499312(CHEMBL3735271)
Affinity DataKi: >6.00E+4nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499317(CHEMBL3735043)
Affinity DataKi: >6.00E+4nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499313(CHEMBL3735387)
Affinity DataKi: >6.00E+4nMAssay Description:Competition binding affinity to MDMX (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed