Affinity DataIC50: 18nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 2.15E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 2.24E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.65E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.21E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 7.37E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+3nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at human platelet P2Y1 receptor assessed as inhibition of ADP-induced increase in cytosolic calcium level by FLUO-4 staining base...More data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+5nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Antagonist activity at human platelet P2Y12 receptor assessed as inhibition of ADP-mediated decrease in intra-platelet phosphorylated VASP by FLUO-4 ...More data for this Ligand-Target Pair
Affinity DataIC50: <2.50E+5nMAssay Description:Partial antagonist activity at human platelet P2Y12 receptor assessed as inhibition of PGE1/ADP-mediated decrease in intra-platelet phosphorylated VA...More data for this Ligand-Target Pair