Compile Data Set for Download or QSAR
maximum 50k data
Found 69 Enz. Inhib. hit(s) with all data for entry = 50006456
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499996(CHEMBL3740019)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500007(CHEMBL3742276)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500011(CHEMBL3739533)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500011(CHEMBL3739533)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500006(CHEMBL3742253)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500013(CHEMBL3740558)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499999(CHEMBL3742198)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499998(CHEMBL3739762)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500006(CHEMBL3742253)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499996(CHEMBL3740019)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500015(CHEMBL3741318)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500003(CHEMBL3742103)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500003(CHEMBL3742103)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500010(CHEMBL3740351)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500003(CHEMBL3742103)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500016(CHEMBL3740874)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500001(CHEMBL3741483)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499998(CHEMBL3739762)
Affinity DataIC50:  36nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499999(CHEMBL3742198)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500007(CHEMBL3742276)
Affinity DataIC50:  46nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500011(CHEMBL3739533)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...)
Affinity DataIC50:  55nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500014(CHEMBL3741260)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500006(CHEMBL3742253)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500014(CHEMBL3741260)
Affinity DataIC50:  89nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499997(CHEMBL3741161)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500017(CHEMBL3739505)
Affinity DataIC50:  96nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500015(CHEMBL3741318)
Affinity DataIC50:  101nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500012(CHEMBL3739900)
Affinity DataIC50:  116nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500002(CHEMBL3740847)
Affinity DataIC50:  122nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500013(CHEMBL3740558)
Affinity DataIC50:  122nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500016(CHEMBL3740874)
Affinity DataIC50:  128nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500008(CHEMBL3741658)
Affinity DataIC50:  151nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500005(CHEMBL3739542)
Affinity DataIC50:  164nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499998(CHEMBL3739762)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500007(CHEMBL3742276)
Affinity DataIC50:  199nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500009(CHEMBL3740042)
Affinity DataIC50:  228nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500002(CHEMBL3740847)
Affinity DataIC50:  229nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500010(CHEMBL3740351)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500005(CHEMBL3739542)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499996(CHEMBL3740019)
Affinity DataIC50:  344nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500005(CHEMBL3739542)
Affinity DataIC50:  384nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500000(CHEMBL3739513)
Affinity DataIC50:  406nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500010(CHEMBL3740351)
Affinity DataIC50:  433nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50499997(CHEMBL3741161)
Affinity DataIC50:  493nMAssay Description:Antagonist activity at adrenergic alpha1D receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500001(CHEMBL3741483)
Affinity DataIC50:  552nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...)
Affinity DataIC50:  555nMAssay Description:Antagonist activity at adrenergic alpha1A receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)-1-piperazinyl]-3-(1-naphtha...)
Affinity DataIC50:  634nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500002(CHEMBL3740847)
Affinity DataIC50:  684nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50500014(CHEMBL3741260)
Affinity DataIC50:  769nMAssay Description:Antagonist activity at adrenergic alpha1B receptor (unknown origin) by firefly and renilla dual glo luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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