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Found 44 Enz. Inhib. hit(s) with all data for entry = 50046963
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140134(CHEMBL3753869)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140131(CHEMBL3752249)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140083(CHEMBL3752210)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140135(CHEMBL3753379)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of ASCT2 (unknown origin)-mediated glutamine transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140127(CHEMBL3754498)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140127(CHEMBL3754498)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140083(CHEMBL3752210)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140081(CHEMBL3752103)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140133(CHEMBL3753592)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140122(CHEMBL3754053)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140122(CHEMBL3754053)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140129(CHEMBL3752700)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140082(CHEMBL3754059)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140130(CHEMBL3752483)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140133(CHEMBL3753592)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140125(CHEMBL3753808)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140082(CHEMBL3754059)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140080(CHEMBL3754415)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140084(CHEMBL3753993)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140079(CHEMBL3753404)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140126(CHEMBL3752316)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140124(CHEMBL3754369)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140079(CHEMBL3753404)
Affinity DataIC50:  2.25E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140132(CHEMBL3752943)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140123(CHEMBL3753173)
Affinity DataIC50:  2.56E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140132(CHEMBL3752943)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140136(CHEMBL3576945)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of ASCT2 (unknown origin)-mediated glutamine transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140124(CHEMBL3754369)
Affinity DataIC50:  3.37E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140131(CHEMBL3752249)
Affinity DataIC50:  3.38E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140130(CHEMBL3752483)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140126(CHEMBL3752316)
Affinity DataIC50:  4.01E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140123(CHEMBL3753173)
Affinity DataIC50:  4.17E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140081(CHEMBL3752103)
Affinity DataIC50:  4.83E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140125(CHEMBL3753808)
Affinity DataIC50:  5.08E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140134(CHEMBL3753869)
Affinity DataIC50:  5.72E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140128(CHEMBL3752494)
Affinity DataIC50:  5.96E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140128(CHEMBL3752494)
Affinity DataIC50:  6.82E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140080(CHEMBL3754415)
Affinity DataIC50:  6.91E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088537(CHEMBL6251 | US10189805, Compound 1)
Affinity DataIC50:  7.02E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmino acid transporter(Rattus norvegicus)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140084(CHEMBL3753993)
Affinity DataIC50:  8.64E+4nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50140129(CHEMBL3752700)
Affinity DataIC50:  1.42E+5nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088534(CHEMBL3576929 | US10189805, Compound 5)
Affinity DataIC50:  3.12E+5nMAssay Description:Inhibition of ASCT2 (unknown origin)-mediated glutamine transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088537(CHEMBL6251 | US10189805, Compound 1)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of ASCT2 (unknown origin)-mediated glutamine transportMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral amino acid transporter B(0)(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088537(CHEMBL6251 | US10189805, Compound 1)
Affinity DataIC50:  1.20E+6nMAssay Description:Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed