TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 173nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 239nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 325nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 347nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 359nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 381nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 403nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 549nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 591nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 653nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataIC50: 783nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair