Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 7325
TargetAurora kinase B(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

LigandPNGBDBM189379(5-O-ethyl 3-O-methyl 4-(2,3-dichlorophenyl)-2,6-di...)
Affinity DataKd:  1.14E+3nMpH: 8.0 T: 2°CAssay Description:Calorimetric titrations were performed in a Microcal iTC 200 microcalorimeter. Freshly purified 5 µM protein (Aurora A/B kinases) was titrated agains...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

LigandPNGBDBM189380(5-methyl-4-(2-thiazolylazo)resorcinol | PTK66)
Affinity DataKd:  500nMpH: 8.0 T: 2°CAssay Description:Calorimetric titrations were performed in a Microcal iTC 200 microcalorimeter. Freshly purified 5 µM protein (Aurora A/B kinases) was titrated agains...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

LigandPNGBDBM189380(5-methyl-4-(2-thiazolylazo)resorcinol | PTK66)
Affinity DataKd:  1.75E+3nMpH: 8.0 T: 2°CAssay Description:Calorimetric titrations were performed in a Microcal iTC 200 microcalorimeter. Freshly purified 5 µM protein (Aurora A/B kinases) was titrated agains...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed