Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50047280
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50161830(CHEMBL3793439)
Affinity DataIC50:  10nMAssay Description:Inhibition of HDAC4 catalytic domain (unknown origin) using Boc-Lys(TFA)-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50160874(CHEMBL3794485 | US9505736, (1S,2S,3S)-2-(4-(5- (Di...)
Affinity DataIC50:  30nMAssay Description:Inhibition of HDAC4 catalytic domain (unknown origin) using Boc-Lys(TFA)-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50161829(CHEMBL3794140)
Affinity DataIC50:  40nMAssay Description:Inhibition of HDAC4 catalytic domain (unknown origin) using Boc-Lys(TFA)-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50161831(CHEMBL3793932 | US9505736, (1S,2S,3S)-1-Fluoro-N-h...)
Affinity DataIC50:  40nMAssay Description:Inhibition of HDAC4 catalytic domain (unknown origin) using Boc-Lys(TFA)-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50160875(CHEMBL3794334 | US9765054, Compound 50d)
Affinity DataIC50:  80nMAssay Description:Inhibition of HDAC4 catalytic domain (unknown origin) using Boc-Lys(TFA)-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50160873(CHEMBL3794544 | US9765054, Compound 50j)
Affinity DataIC50:  140nMAssay Description:Inhibition of HDAC4 catalytic domain (unknown origin) using Boc-Lys(TFA)-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50160874(CHEMBL3794485 | US9505736, (1S,2S,3S)-2-(4-(5- (Di...)
Affinity DataIC50:  150nMAssay Description:Inhibition of HDAC4 in human Jurkat E6-1 cells using Lys-TFA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50161829(CHEMBL3794140)
Affinity DataIC50:  230nMAssay Description:Inhibition of HDAC4 in human Jurkat E6-1 cells using Lys-TFA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50160873(CHEMBL3794544 | US9765054, Compound 50j)
Affinity DataIC50:  430nMAssay Description:Inhibition of HDAC4 in human Jurkat E6-1 cells using Lys-TFA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50155843(CHEMBL3793034 | US9765054, Compound 50K)
Affinity DataIC50:  510nMAssay Description:Inhibition of HDAC4 in human Jurkat E6-1 cells using Lys-TFA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50155804(CHEMBL3793569)
Affinity DataIC50:  730nMAssay Description:Inhibition of HDAC4 in human Jurkat E6-1 cells using Lys-TFA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50155803(CHEMBL3793455 | US9505736, (1S,2S,3S)-1-Chloro-N-h...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of HDAC4 in human Jurkat E6-1 cells using Lys-TFA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Biofocus

Curated by ChEMBL
LigandPNGBDBM50160879(CHEMBL3793392 | US9505736, (1S,2S,3S)-1-Fluoro-2-(...)
Affinity DataKd:  20nMAssay Description:Binding affinity to HDAC4 catalytic domain (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair