Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 50047139
TargetKallikrein-2(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  1.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  3.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human tissue kallikrein-5 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human tissue kallikrein-3 expressed in baculovirus infected insect cells using Abz-KLYSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-6(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of human tissue kallikrein-6 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Campus

Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human tissue kallikrein-7 expressed in baculovirus infected insect cells using Abz-KLYSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed