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Found 25 Enz. Inhib. hit(s) with all data for entry = 50047287
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157866(CHEMBL3785238)
Affinity DataKi:  16nMAssay Description:Tested for neuronal nicotinic acetylcholine receptor (nAChR) binding in a whole rat brain preparation using [3H]-cystine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157867(CHEMBL3786384)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157858(CHEMBL3786154)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157875(CHEMBL3786776)
Affinity DataKi:  26nMAssay Description:Tested for functional activity against neuronal nicotinic acetylcholine receptor(nAChR) expressed in K177 cells using isotopic rubidium efflux assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157876(CHEMBL3787276)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157865(CHEMBL3786829)
Affinity DataKi:  29nMAssay Description:Tested for neuronal nicotinic acetylcholine receptor (nAChR) binding in a whole rat brain preparation using [3H]-cystine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157869(CHEMBL3785368)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157868(CHEMBL3786998)
Affinity DataKi:  32nMAssay Description:Tested for functional activity against neuronal nicotinic acetylcholine receptor(nAChR) expressed in K177 cells using isotopic rubidium efflux assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50034168(CHEMBL3359231)
Affinity DataKi:  44nMAssay Description:Tested for neuronal nicotinic acetylcholine receptor (nAChR) binding in a whole rat brain preparation using [3H]-cystine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50034167(CHEMBL3359232)
Affinity DataKi:  59nMAssay Description:Tested for neuronal nicotinic acetylcholine receptor (nAChR) binding in a whole rat brain preparation using [3H]-cystine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157874(CHEMBL3786813)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157813(CHEMBL3786259)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157871(CHEMBL3786461)
Affinity DataKi:  103nMAssay Description:Tested for functional activity against neuronal nicotinic acetylcholine receptor(nAChR) expressed in K177 cells using isotopic rubidium efflux assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50034164(CHEMBL3352885)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157810(CHEMBL3787269)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157873(CHEMBL3786729)
Affinity DataKi:  121nMAssay Description:Tested for functional activity against neuronal nicotinic acetylcholine receptor(nAChR) expressed in K177 cells using isotopic rubidium efflux assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157812(CHEMBL3787434)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50034165(CHEMBL3359233)
Affinity DataKi:  139nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157811(CHEMBL3786949)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157872(CHEMBL3786283)
Affinity DataKi:  189nMAssay Description:Tested for functional activity against neuronal nicotinic acetylcholine receptor(nAChR) expressed in K177 cells using isotopic rubidium efflux assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157814(CHEMBL3787177)
Affinity DataKi:  238nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157815(CHEMBL3785416)
Affinity DataKi:  354nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157870(CHEMBL3786749)
Affinity DataKi: >2.00E+3nMAssay Description:Tested for neuronal nicotinic acetylcholine receptor (nAChR) binding in a whole rat brain preparation using [3H]-cystine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157877(CHEMBL3785243)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Renmin Hospital Of Wuhan University

Curated by ChEMBL
LigandPNGBDBM50157855(CHEMBL3785134)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed