Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50047232
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155330BDBM50155330(CHEMBL3781890)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155326BDBM50155326(CHEMBL3780463)
Affinity DataIC50: 680nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155332BDBM50155332(CHEMBL3781465)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155329BDBM50155329(CHEMBL3779912)
Affinity DataIC50: 820nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155324BDBM50155324(CHEMBL3780894)
Affinity DataIC50: 850nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155328BDBM50155328(CHEMBL3781727)
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155325BDBM50155325(CHEMBL3780991)
Affinity DataIC50: 4.60E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155323BDBM50155323(CHEMBL3781370)
Affinity DataIC50: 6.86E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155331BDBM50155331(CHEMBL3781952)
Affinity DataIC50: 7.65E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155448BDBM50155448(CHEMBL3781901)
Affinity DataIC50: 8.80E+3nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universit£&Quot;G. D'Annunzio&Quot

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155327BDBM50155327(CHEMBL3781940)
Affinity DataIC50: 1.08E+5nMAssay Description:Antagonist activity at PPARalpha (unknown origin) expressed in HEK293A cells assessed as inhibition of GW7647-induced transactivation after 16 to 18 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed