Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50047590
LigandPNGBDBM50177043(CHEMBL3814671)
Affinity DataIC50:  339nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177042(CHEMBL3730906)
Affinity DataIC50:  427nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50177033(CHEMBL3813839)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human PI3Kgamma using PIP2 as substrate by HTRF assay in presence of biotin-PIP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177041(CHEMBL3814491)
Affinity DataIC50:  2.46E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50429613(CHEMBL2334590)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177040(CHEMBL3814642)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177039(CHEMBL3814308)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177038(CHEMBL3814655)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50177032(CHEMBL3814407)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human PI3Kgamma using PIP2 as substrate by HTRF assay in presence of biotin-PIP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50177031(CHEMBL3814969)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of human PI3Kgamma using PIP2 as substrate by HTRF assay in presence of biotin-PIP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50177044(CHEMBL3814695)
Affinity DataIC50:  6.17E+3nMAssay Description:Inhibition of human PI3Kgamma using PIP2 as substrate by HTRF assay in presence of biotin-PIP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177037(CHEMBL3814438)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177036(CHEMBL1528007)
Affinity DataIC50:  6.92E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50177045(CHEMBL3814733)
Affinity DataIC50:  6.92E+3nMAssay Description:Inhibition of human PI3Kgamma using PIP2 as substrate by HTRF assay in presence of biotin-PIP3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177035(CHEMBL3814774)
Affinity DataIC50:  8.13E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50177034(CHEMBL3813732)
Affinity DataIC50:  8.51E+3nMAssay Description:Inhibition of human full length recombinant His-tagged PIK3CD/PIK3R1 expressed in baculovirus expression system after 60 mins by LanthaScreen Eu bind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed