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Found 13 Enz. Inhib. hit(s) with all data for entry = 50047757
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187704(CHEMBL3828024)
Affinity DataIC50:  25nMAssay Description:Inhibition of PSMA (unknown origin) assessed as reduction in glutamate formation using NAAG as substrate preincubated for 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187705(CHEMBL3828668)
Affinity DataIC50:  28nMAssay Description:Inhibition of PSMA (unknown origin) assessed as reduction in glutamate formation using NAAG as substrate preincubated for 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50106240(6-Chloro-2-(2-hydroxy-biphenyl-3-yl)-1H-indole-5-c...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187705(CHEMBL3828668)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187711(CHEMBL3827463)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187707(CHEMBL3827292)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187708(CHEMBL3827374)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187709(CHEMBL3827645)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187710(CHEMBL3827788)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187706(CHEMBL3828589)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187713(CHEMBL3828730)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50102768(2-(2-Hydroxy-phenyl)-1H-indole-5-carboxamidine | C...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50187712(CHEMBL3828185)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed