Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50047711
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50185129(CHEMBL3822808)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-hU2 from human UT2 receptor expressed in CHO cells after 90 mins by gamma counter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50185139(CHEMBL3823939)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-hU2 from human UT2 receptor expressed in CHO cells after 90 mins by gamma counter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50185136(CHEMBL3823122)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-hU2 from human UT2 receptor expressed in CHO cells after 90 mins by gamma counter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50185137(CHEMBL3823569)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-hU2 from human UT2 receptor expressed in CHO cells after 90 mins by gamma counter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50185135(CHEMBL3823484)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-hU2 from human UT2 receptor expressed in CHO cells after 90 mins by gamma counter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50185138(CHEMBL3822950)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-hU2 from human UT2 receptor expressed in CHO cells after 90 mins by gamma counter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185135(CHEMBL3823484)
Affinity DataEC50:  7.90nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for URP -induced aortic contractions at 10'-5M relati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185136(CHEMBL3823122)
Affinity DataEC50:  9.5nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for URP -induced aortic contractions at 10'-5M relati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185137(CHEMBL3823569)
Affinity DataEC50:  9.10nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for URP -induced aortic contractions at 10'-5M relati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185139(CHEMBL3823939)
Affinity DataEC50:  3.70nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for URP -induced aortic contractions at 10'-5M relati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185138(CHEMBL3822950)
Affinity DataEC50:  4.80nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185138(CHEMBL3822950)
Affinity DataEC50:  3.5nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for URP -induced aortic contractions at 10'-5M relati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185135(CHEMBL3823484)
Affinity DataEC50:  5nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185136(CHEMBL3823122)
Affinity DataEC50:  15nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185137(CHEMBL3823569)
Affinity DataEC50:  2.60nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185139(CHEMBL3823939)
Affinity DataEC50:  1.60nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185129(CHEMBL3822808)
Affinity DataEC50:  13nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for URP -induced aortic contractions at 10'-5M relati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50185129(CHEMBL3822808)
Affinity DataEC50:  9.5nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed