Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50047449
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168058(CHEMBL3798461)
Affinity DataIC50:  110nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168056(CHEMBL3799363)
Affinity DataIC50:  250nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50123151(CHEMBL3623223)
Affinity DataIC50:  470nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168057(CHEMBL3800417)
Affinity DataIC50:  530nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed