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Found 6 Enz. Inhib. hit(s) with all data for entry = 50048037
TargetCell division protein FtsZ(Staphylococcus aureus)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50079356(CHEMBL511201)
Affinity DataIC50:  154nMAssay Description:Inhibition of Staphylococcus aureus FtsZ GTPase activityMore data for this Ligand-Target Pair
TargetCell division protein FtsZ(Escherichia coli)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50203126(3,4-dimethoxy-6,7-dihydro-[1,3]dioxolo[4,5-g]pyrid...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant Escherichia coli K12 FtsZ assembly by light-scattering assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division protein FtsZ(Escherichia coli)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50203126(3,4-dimethoxy-6,7-dihydro-[1,3]dioxolo[4,5-g]pyrid...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of recombinant Escherichia coli K12 FtsZ GTPase activity by malachite green sodium molybdate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division protein FtsZ(Staphylococcus aureus)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50201769(CHEMBL3416823)
Affinity DataIC50:  3.75E+4nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 N-terminal His6-tagged FtsZ GTPase activity expressed in Escherichia coli BL21(DE3) assessed as reduct...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division protein FtsZ(Staphylococcus aureus)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50320891(9-O-[3-(4-Chloro-phenoxyl)propyl]-berberine bromid...)
Affinity DataIC50:  7.74E+4nMAssay Description:Inhibition of Staphylococcus aureus N-terminal His6-tagged FtsZ GTPase activity expressed in Escherichia coli BL21(DE3) preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division protein FtsZ(Staphylococcus aureus)
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50201768(CHEMBL2413354)
Affinity DataIC50:  3.17E+5nMAssay Description:Inhibition of Staphylococcus aureus ATCC 29213 N-terminal His6-tagged FtsZ GTPase activity expressed in Escherichia coli BL21(DE3) assessed as reduct...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed