Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50047564
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175036BDBM50175036(CHEMBL3809599)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175039BDBM50175039(CHEMBL3808639)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175038BDBM50175038(CHEMBL3810162)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175064BDBM50175064(CHEMBL3809530)
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175041BDBM50175041(CHEMBL3809034)
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175035BDBM50175035(CHEMBL3808866)
Affinity DataIC50: 330nMAssay Description:Inhibition of human HDAC3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175037BDBM50175037(CHEMBL3808986)
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175063BDBM50175063(CHEMBL3808977)
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175060BDBM50175060(CHEMBL3809171)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175044BDBM50175044(CHEMBL3809231)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175040BDBM50175040(CHEMBL3810111)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175035BDBM50175035(CHEMBL3808866)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175045BDBM50175045(CHEMBL3808864)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175067BDBM50175067(CHEMBL3809999)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175066BDBM50175066(CHEMBL3810053)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175046BDBM50175046(CHEMBL3809931)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175043BDBM50175043(CHEMBL3809454)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175065BDBM50175065(CHEMBL3808426)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175062BDBM50175062(CHEMBL3810196)
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175061BDBM50175061(CHEMBL3809732)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175047BDBM50175047(CHEMBL3809504)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175048BDBM50175048(CHEMBL3810335)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175042BDBM50175042(CHEMBL3810397)
Affinity DataIC50: 2.39E+4nMAssay Description:Inhibition of recombinant human His-tagged HDAC1 expressed in insect cells preincubated for 10 mins followed by addition of FLUOR DE LYS as fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Irbm Science Park

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50175035BDBM50175035(CHEMBL3808866)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/13/2017
Entry Details Article
PubMed