Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50047568
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175290(CHEMBL3810385)
Affinity DataIC50:  67nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175288(CHEMBL3809413)
Affinity DataIC50:  130nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175289(CHEMBL3810032)
Affinity DataIC50:  900nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175293(CHEMBL3808576)
Affinity DataIC50:  910nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPsychosine receptor(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175290(CHEMBL3810385)
Affinity DataIC50: >1.00E+4nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged TDAG8 receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP res...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175294(CHEMBL3727521)
Affinity DataIC50: >1.00E+4nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOvarian cancer G-protein coupled receptor 1(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175290(CHEMBL3810385)
Affinity DataIC50: >1.00E+4nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged OGR1 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent nuclear factor of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175291(CHEMBL3809249)
Affinity DataIC50: >1.00E+4nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 4(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50175292(CHEMBL3810150)
Affinity DataIC50: >1.00E+4nMpH: 7.2Assay Description:Antagonist activity at N-terminal HA-tagged GPR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent cAMP response elem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed