Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 4758
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81963(CHOLECYSTOKININ | CCK33 | CAS_9011-97-6 | CCK)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81963(CHOLECYSTOKININ | CCK33 | CAS_9011-97-6 | CCK)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81964(NSC_5486814 | CAS_5486814 | Neuromedin C | Gastrin)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81962(S-L-365,260)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81964(NSC_5486814 | CAS_5486814 | Neuromedin C | Gastrin)
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005459(CHEMBL9485 | CR 1409 | 4-(3,4-Dichloro-benzoylamin...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Dog)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Dog)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  39nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  151nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  250nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Dog)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81964(NSC_5486814 | CAS_5486814 | Neuromedin C | Gastrin)
Affinity DataKi:  560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50061220(CHEMBL70380 | L-365,260 | 1-(1-Methyl-2-oxo-5-phen...)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005459(CHEMBL9485 | CR 1409 | 4-(3,4-Dichloro-benzoylamin...)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetCholecystokinin(Pig)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005459(CHEMBL9485 | CR 1409 | 4-(3,4-Dichloro-benzoylamin...)
Affinity DataKi:  2.20E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed