Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50047793
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190178(CHEMBL3828321)
Affinity DataIC50:  72nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190311(CHEMBL3828131)
Affinity DataIC50:  76nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190176(CHEMBL3828240)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190171(CHEMBL3827219)
Affinity DataIC50:  92nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190177(CHEMBL3828609)
Affinity DataIC50:  105nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190184(CHEMBL3827727)
Affinity DataIC50:  107nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190314(CHEMBL3827511)
Affinity DataIC50:  122nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190175(CHEMBL3828624)
Affinity DataIC50:  124nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190170(CHEMBL3827901)
Affinity DataIC50:  131nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190313(CHEMBL3828006)
Affinity DataIC50:  134nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190179(CHEMBL3828098)
Affinity DataIC50:  135nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190315(CHEMBL3827702)
Affinity DataIC50:  145nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190174(CHEMBL3827726)
Affinity DataIC50:  148nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190310(CHEMBL3827844)
Affinity DataIC50:  151nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190316(CHEMBL3828407)
Affinity DataIC50:  157nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190180(CHEMBL3827895)
Affinity DataIC50:  157nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190312(CHEMBL3828350)
Affinity DataIC50:  173nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190257(CHEMBL3828150)
Affinity DataIC50:  184nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190169(CHEMBL3828114)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190173(CHEMBL3828491)
Affinity DataIC50:  205nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190185(CHEMBL3827240)
Affinity DataIC50:  293nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190172(CHEMBL3828571)
Affinity DataIC50:  379nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190183(CHEMBL3828352)
Affinity DataIC50:  406nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190181(CHEMBL3827724)
Affinity DataIC50:  561nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50190182(CHEMBL3828397)
Affinity DataIC50:  582nMAssay Description:Inhibition of recombinant human N-terminal His-tagged GSK-3beta expressed in Escherichia coli using glycogen synthase-2 as substrate and ATP measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed