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Found 5 Enz. Inhib. hit(s) with all data for entry = 50048048
TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
Rytmion

Curated by ChEMBL
LigandPNGBDBM50202477(CHEMBL3955249)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of GTPgammaS-induced activation of GIRK1/4 (unknown origin) expressed in HEK293 cells assessed as decrease in channel current after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
Rytmion

Curated by ChEMBL
LigandPNGBDBM50202479(CHEBI:69714 | Euphorbiaproliferin C)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of GTPgammaS-induced activation of GIRK1/4 (unknown origin) expressed in HEK293 cells assessed as decrease in channel current after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
Rytmion

Curated by ChEMBL
LigandPNGBDBM50202481(CHEMBL3901192)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of GTPgammaS-induced activation of GIRK1/4 (unknown origin) expressed in HEK293 cells assessed as decrease in channel current after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
Rytmion

Curated by ChEMBL
LigandPNGBDBM50202478(CHEMBL3899370)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of GTPgammaS-induced activation of GIRK1/4 (unknown origin) expressed in HEK293 cells assessed as decrease in channel current after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
Rytmion

Curated by ChEMBL
LigandPNGBDBM50202480(CHEMBL3961215)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of GTPgammaS-induced activation of GIRK1/4 (unknown origin) expressed in HEK293 cells assessed as decrease in channel current after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed