Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50048178
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50103521(CHEBI:8228 | Actos | Duetact | Pioglitazone | US20...)
Affinity DataEC50:  500nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in African green monkey COS7 cells after 42 hrs by dual luciferase repo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207273(CHEMBL3891909)
Affinity DataEC50:  600nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataEC50:  700nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50103521(CHEBI:8228 | Actos | Duetact | Pioglitazone | US20...)
Affinity DataEC50:  1.60E+3nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207276(CHEMBL3973020)
Affinity DataEC50:  2.10E+3nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207272(CHEMBL3960906)
Affinity DataEC50:  2.80E+3nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207274(CHEMBL3962023)
Affinity DataEC50:  3.10E+3nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207273(CHEMBL3891909)
Affinity DataEC50:  3.40E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in African green monkey COS7 cells after 42 hrs by dual luciferase repo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataEC50:  4.70E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in African green monkey COS7 cells after 42 hrs by dual luciferase repo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207275(CHEMBL3913928)
Affinity DataEC50:  5.40E+3nMAssay Description:Displacement of Fluoromone from GST-tagged recombinant human PPARgamma ligand binding domain by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50207272(CHEMBL3960906)
Affinity DataEC50:  2.17E+4nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in African green monkey COS7 cells after 42 hrs by dual luciferase repo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed