Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50048151
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206448(CHEMBL3944542)
Affinity DataIC50:  2.94E+4nMAssay Description:Inhibition of 5-FAM-DPPLHSpTAI-OH binding to PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) after 1 hr by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206451(CHEMBL3894239)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of 5-FAM-DPPLHSpTAI-OH binding to PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) after 1 hr by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206451(CHEMBL3894239)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of full-length PLK1 (unknown origin) expressed in Escherichia coli Rosetta (DE3) using ALMDASFADQ as substrate after 40 mins by fluorimetr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206448(CHEMBL3944542)
Affinity DataKd:  1.05E+4nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206455(CHEMBL3922258)
Affinity DataKd:  6.90E+3nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206449(CHEMBL3944679)
Affinity DataKd:  5.10E+3nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50005003(CHEMBL2392423)
Affinity DataKd:  6.88E+4nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206452(CHEMBL3908343)
Affinity DataKd:  7.37E+4nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206453(CHEMBL3978761)
Affinity DataKd:  6.43E+4nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206454(CHEMBL3928373)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206450(CHEMBL3921162)
Affinity DataKd:  5.60E+3nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50206451(CHEMBL3894239)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to NT-647 labeled PLK1 polo-box domain (unknown origin) expressed in Escherichia coli Rosetta (DE3) by microscale thermophoresis bas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed