Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50009968
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM59542(SMR000523991 | cid_1088438 | MLS001201458 | 1-(4-m...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533841(CHEMBL4472193)
Affinity DataIC50: 5.74E+3nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533841(CHEMBL4472193)
Affinity DataIC50: 6.45E+3nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM62334(1-[(4-chlorophenyl)methyl]benzimidazol-2-amine | c...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533839(CHEMBL4474194)
Affinity DataIC50: 7.78E+3nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533839(CHEMBL4474194)
Affinity DataIC50: 9.04E+3nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533838(CHEMBL4586513)
Affinity DataIC50: 9.22E+3nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM62334(1-[(4-chlorophenyl)methyl]benzimidazol-2-amine | c...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533838(CHEMBL4586513)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533837(CHEMBL4462798)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533835(CHEMBL4451566)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533836(CHEMBL4534055)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533837(CHEMBL4462798)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533840(CHEMBL378112)
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of human NOD1 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533840(CHEMBL378112)
Affinity DataIC50: 2.34E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533836(CHEMBL4534055)
Affinity DataIC50: 2.46E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50533835(CHEMBL4451566)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM59542(SMR000523991 | cid_1088438 | MLS001201458 | 1-(4-m...)
Affinity DataIC50: 5.49E+4nMAssay Description:Inhibition of human NOD2 over-expressed in HEK-Blue cells assessed as inhibition of C12-iE-DAP induced NF-kappaB transcriptional activity preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed