Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50047833
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 0.220nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192811BDBM50192811(CHEMBL3971502)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192807BDBM50192807(CHEMBL3984947)
Affinity DataIC50: 0.360nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of hypotonicity-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192804BDBM50192804(CHEMBL3933401)
Affinity DataIC50: 0.570nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192820BDBM50192820(CHEMBL3950646)
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192808BDBM50192808(CHEMBL3915150)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192779BDBM50192779(CHEMBL3957347)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192817BDBM50192817(CHEMBL3924485)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192781BDBM50192781(CHEMBL3985107)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192827BDBM50192827(CHEMBL3985405)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of hypotonicity-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192826BDBM50192826(CHEMBL3979114)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192803BDBM50192803(CHEMBL3906685)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192819BDBM50192819(CHEMBL3908777)
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192822BDBM50192822(CHEMBL3897222)
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192776BDBM50192776(CHEMBL3979627)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192778BDBM50192778(CHEMBL3942384)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192816BDBM50192816(CHEMBL3968344)
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192828BDBM50192828(CHEMBL3914089)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192824BDBM50192824(CHEMBL3924665)
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192774BDBM50192774(CHEMBL3986034)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192813BDBM50192813(CHEMBL3896628)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192777BDBM50192777(CHEMBL3915675)
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192825BDBM50192825(CHEMBL3976867)
Affinity DataIC50: 8.40nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 8.60nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192804BDBM50192804(CHEMBL3933401)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192811BDBM50192811(CHEMBL3971502)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192807BDBM50192807(CHEMBL3984947)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192823BDBM50192823(CHEMBL3906074)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192815BDBM50192815(CHEMBL3906180)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192820BDBM50192820(CHEMBL3950646)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192810BDBM50192810(CHEMBL3942090)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192802BDBM50192802(CHEMBL3927993)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192779BDBM50192779(CHEMBL3957347)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192775BDBM50192775(CHEMBL3915493)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192772BDBM50192772(CHEMBL3967702)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192806BDBM50192806(CHEMBL3960867)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192780BDBM50192780(CHEMBL3977334)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192817BDBM50192817(CHEMBL3924485)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192822BDBM50192822(CHEMBL3897222)
Affinity DataIC50: 57nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192821BDBM50192821(CHEMBL2133556)
Affinity DataIC50: 57nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192828BDBM50192828(CHEMBL3914089)
Affinity DataIC50: 57nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192814BDBM50192814(CHEMBL3933578)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192778BDBM50192778(CHEMBL3942384)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192824BDBM50192824(CHEMBL3924665)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192813BDBM50192813(CHEMBL3896628)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192777BDBM50192777(CHEMBL3915675)
Affinity DataIC50: 290nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192802BDBM50192802(CHEMBL3927993)
Affinity DataIC50: 360nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192776BDBM50192776(CHEMBL3979627)
Affinity DataIC50: 410nMAssay Description:Antagonist activity at rat TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
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