TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 105nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 106nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 192nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 262nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 273nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 565nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain MAO-A using [14C]5-HT as substrate preincubated for 20 mins followed by substrate addition measured after 5 mi...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 3.52E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 3.65E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 6.46E+3nMAssay Description:Binding affinity for protein kinase C-alpha C1a and C1b domainsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Binding affinity for protein kinase C-alpha C1a and C1b domainsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 6.63E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 7.59E+3nMAssay Description:Binding affinity for protein kinase C-alpha C1a and C1b domainsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 8.78E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 9.36E+3nMAssay Description:Binding affinity for protein kinase C-alpha C1a and C1b domainsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
North-West University
Curated by ChEMBL
North-West University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate by fluorescence spectrophotometryMore data for this Ligand-Target Pair