Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50048186
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataKi:  9.80E+3nMAssay Description:Competitive inhibition of porcine pancreatic lipase 4-nitrophenyl butyrate substrate preincubated for 30 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207386(CHEMBL3967165)
Affinity DataKi:  1.75E+4nMAssay Description:Competitive inhibition of porcine pancreatic lipase 4-nitrophenyl butyrate substrate preincubated for 30 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207381(CHEMBL3934940)
Affinity DataKi:  1.96E+4nMAssay Description:Competitive inhibition of porcine pancreatic lipase 4-nitrophenyl butyrate substrate preincubated for 30 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207370(CHEMBL3896540)
Affinity DataKi:  2.16E+4nMAssay Description:Competitive inhibition of porcine pancreatic lipase 4-nitrophenyl butyrate substrate preincubated for 30 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  990nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207386(CHEMBL3967165)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207381(CHEMBL3934940)
Affinity DataIC50:  8.72E+3nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207370(CHEMBL3896540)
Affinity DataIC50:  9.58E+3nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207390(CHEMBL3976270)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207395(CHEMBL3908464)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207371(CHEMBL3979181)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207379(CHEMBL3944368)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207388(CHEMBL3906649)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207373(CHEMBL3931385)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207394(CHEMBL3906497)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207385(CHEBI:6646 | Mahanimbine | Rel-(+)-Mahanimbine)
Affinity DataIC50:  1.79E+4nMAssay Description:Inhibition of pancreatic lipase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207376(CHEMBL3932922)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207393(CHEMBL3905980)
Affinity DataIC50:  1.99E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207378(CHEMBL3977704)
Affinity DataIC50:  2.31E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207387(CHEMBL3897958)
Affinity DataIC50:  2.31E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207396(CHEMBL3977167)
Affinity DataIC50:  2.42E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207382(CHEMBL3945483)
Affinity DataIC50:  2.66E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207380(CHEMBL3931968)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207375(CHEMBL3982037)
Affinity DataIC50:  2.94E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207389(CHEMBL3985837)
Affinity DataIC50:  2.97E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207377(CHEMBL3911394)
Affinity DataIC50:  3.28E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207392(CHEMBL3957164)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207391(CHEMBL3966764)
Affinity DataIC50:  3.62E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207372(CHEMBL3948881)
Affinity DataIC50:  4.41E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Sus scrofa (Pig))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207374(CHEMBL3915474)
Affinity DataIC50:  5.62E+4nMAssay Description:Inhibition of porcine pancreatic lipase assessed as reduction in 4-nitrophenol formation from 4-nitrophenyl butyrate substrate preincubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207384(Koenimbine)
Affinity DataIC50:  1.69E+5nMAssay Description:Inhibition of pancreatic lipase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Birla Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50207383(CHEMBL3893262)
Affinity DataIC50:  4.29E+5nMAssay Description:Inhibition of pancreatic lipase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed