Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50048925
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228785(CHEMBL4060363)
Affinity DataIC50:  0.230nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)
Affinity DataIC50:  0.720nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228779(CHEMBL4074951)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228561(CHEMBL4100369)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228787(CHEMBL4082353)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228818(CHEMBL4103138)
Affinity DataIC50:  12nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228783(CHEMBL4085200)
Affinity DataIC50:  20nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228784(CHEMBL4087240)
Affinity DataIC50:  22nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228788(CHEMBL4087694)
Affinity DataIC50:  23nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228780(CHEMBL4095386)
Affinity DataIC50:  27nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228782(CHEMBL4092943)
Affinity DataIC50:  91nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228786(CHEMBL4065282)
Affinity DataIC50: >100nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50228781(CHEMBL4066344)
Affinity DataIC50: >100nMAssay Description:Inhibition of N-terminal His-tagged full length human recombinant BTK expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Glu, Tyr) pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed