Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50048031
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201680BDBM50201680(CHEMBL3922381)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201693BDBM50201693(CHEMBL3904378)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386790BDBM50386790(CHEMBL1829174 | CHEMBL2047159 | TAK-875 | US119052...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201656BDBM50201656(CHEMBL3966739)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201678BDBM50201678(CHEMBL3896509)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201688BDBM50201688(CHEMBL3923431)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201690BDBM50201690(CHEMBL3889768)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362690BDBM50362690(CHEMBL1829173 | AMG-837)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201689BDBM50201689(CHEMBL3924534)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201681BDBM50201681(CHEMBL3951157)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201682BDBM50201682(CHEMBL3918387)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201694BDBM50201694(CHEMBL3914686)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201696BDBM50201696(CHEMBL3914418)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201685BDBM50201685(CHEMBL3913383)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201686BDBM50201686(CHEMBL3975239)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201695BDBM50201695(CHEMBL3893141)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201670BDBM50201670(CHEMBL3930086)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as induction of IP1 formation after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201679BDBM50201679(CHEMBL3957744)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201670BDBM50201670(CHEMBL3930086)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as induction of intracellular Ca2+ flux preincubated for 40 mins measured for 180 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201687BDBM50201687(CHEMBL3895442)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201683BDBM50201683(CHEMBL3933446)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201691BDBM50201691(CHEMBL3921143)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201684BDBM50201684(CHEMBL3894356)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201677BDBM50201677(CHEMBL3931296)
Affinity DataEC50:  118nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201657BDBM50201657(CHEMBL3905435)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201692BDBM50201692(CHEMBL3964251)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells measured after 18 to 20 hrs by beta-gal based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Rat)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50201670BDBM50201670(CHEMBL3930086)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at GPR40 in rat RINm cells assessed as increase glucose-stimulated insulin secretion after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Rat)
Cadila Healthcare

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50386790BDBM50386790(CHEMBL1829174 | CHEMBL2047159 | TAK-875 | US119052...)
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at GPR40 in rat RINm cells assessed as increase glucose-stimulated insulin secretion after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed