Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50049019
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232960BDBM50232960(CHEMBL4087035)
Affinity DataEC50:  30nMAssay Description:Activation of human CFTR expressed in forskolin-stimulated basolateral membrane permeabilized FRT cells co-expressing YFP assessed as increase in sho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232962BDBM50232962(CHEMBL4079174)
Affinity DataEC50:  31nMAssay Description:Activation of human CFTR expressed in forskolin-stimulated basolateral membrane permeabilized FRT cells co-expressing YFP assessed as increase in sho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232962BDBM50232962(CHEMBL4079174)
Affinity DataEC50:  40nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232960BDBM50232960(CHEMBL4087035)
Affinity DataEC50:  50nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232961BDBM50232961(CHEMBL4097188)
Affinity DataEC50:  120nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232956BDBM50232956(CHEMBL4097536)
Affinity DataEC50:  140nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232967BDBM50232967(CHEMBL4104898)
Affinity DataEC50:  150nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232957BDBM50232957(CHEMBL4080996)
Affinity DataEC50:  160nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232965BDBM50232965(CHEMBL4078552)
Affinity DataEC50:  200nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232949BDBM50232949(CHEMBL4100901)
Affinity DataEC50:  240nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232954BDBM50232954(CHEMBL4096577)
Affinity DataEC50:  500nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232950BDBM50232950(CHEMBL4093184)
Affinity DataEC50:  700nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232951BDBM50232951(CHEMBL4092200)
Affinity DataEC50:  900nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232958BDBM50232958(CHEMBL4067285)
Affinity DataEC50:  900nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232964BDBM50232964(CHEMBL4071412)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232953BDBM50232953(CHEMBL4062768)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232966BDBM50232966(CHEMBL4070362)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232948BDBM50232948(CHEMBL4074144)
Affinity DataEC50:  2.50E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232955BDBM50232955(CHEMBL4070356)
Affinity DataEC50:  2.80E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232959BDBM50232959(CHEMBL4094736)
Affinity DataEC50:  2.80E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232947BDBM50232947(CHEMBL4097540)
Affinity DataEC50:  4.80E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232952BDBM50232952(CHEMBL4084446)
Affinity DataEC50:  5.40E+3nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232963BDBM50232963(CHEMBL4065523)
Affinity DataEC50:  1.80E+4nMAssay Description:Activation of human CFTR expressed in FRT cells co-expressing YFP assessed as increase in forskolin-stimulated iodide influx measured after 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2019
Entry Details Article
PubMed