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Found 12 Enz. Inhib. hit(s) with all data for entry = 50000294
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245492(CHEMBL4082554)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant TACE catalytic domain (unknown origin) using pro-TNFalpha peptide Abz-LAQAVRSSSR-Dpa as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50236621(CHEMBL4078142)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant TACE catalytic domain (unknown origin) using pro-TNFalpha peptide Abz-LAQAVRSSSR-Dpa as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245498(CHEMBL4083562)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant human ASK1 using STK3 peptide as substrate incubated for 30 mins followed by ATP addition measured for 3 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245482(CHEMBL4069275)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245491(CHEMBL4098028)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245499(CHEMBL4085616)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245479(CHEMBL4103552)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245494(CHEMBL4080004)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245481(CHEMBL4060589)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245480(CHEMBL4082477)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled receptor 84(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245516(CHEMBL4090321)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at GPR84 (unknown origin) expressed in cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50245493(CHEMBL4092255)
Affinity DataIC50:  27nMAssay Description:Inhibition of human liver cathepsin B using Boc-Leu-Arg-Arg-AMC as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed