Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50048998
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 20nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50197240(KYS-05080 | N-benzyl-2-(3-(biphenyl-4-yl)-2-(methy...)
Affinity DataKi:  29nMAssay Description:Mixed/noncompetitive inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50197240(KYS-05080 | N-benzyl-2-(3-(biphenyl-4-yl)-2-(methy...)
Affinity DataIC50: 45nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50222222(CHEMBL394956 | N-benzyl-2-(3-(biphenyl-4-yl)-2-((5...)
Affinity DataKi:  51nMAssay Description:Mixed/noncompetitive inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50222222(CHEMBL394956 | N-benzyl-2-(3-(biphenyl-4-yl)-2-((5...)
Affinity DataIC50: 62nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232663(CHEMBL4081075)
Affinity DataIC50: 140nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232638(CHEMBL4084185)
Affinity DataIC50: 240nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232637(CHEMBL4061274)
Affinity DataIC50: 380nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232640(CHEMBL4086668)
Affinity DataIC50: 400nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232637(CHEMBL4061274)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232664(CHEMBL4076211)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232665(CHEMBL4076174)
Affinity DataIC50: 2.04E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232641(CHEMBL4065933)
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232643(CHEMBL3093780)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232644(CHEMBL4067745)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232640(CHEMBL4086668)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232644(CHEMBL4067745)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232642(CHEMBL3093781)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232638(CHEMBL4084185)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50197240(KYS-05080 | N-benzyl-2-(3-(biphenyl-4-yl)-2-(methy...)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232641(CHEMBL4065933)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232639(CHEMBL115066)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232664(CHEMBL4076211)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50148173(N-Benzyl-2-[2-(4-methyl-piperazin-1-yl)-3-phenyl-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232665(CHEMBL4076174)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50148173(N-Benzyl-2-[2-(4-methyl-piperazin-1-yl)-3-phenyl-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of equine serum BCHE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50232642(CHEMBL3093781)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition measured for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed