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Found 10 Enz. Inhib. hit(s) with all data for entry = 50049227
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236985(CHEMBL4098600)
Affinity DataIC50:  310nMAssay Description:Inhibition of human recombinant COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236980(CHEMBL4097499)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236981(CHEMBL4086580)
Affinity DataIC50:  670nMAssay Description:Inhibition of human recombinant COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236984(CHEMBL4069250)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by ADHP pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236985(CHEMBL4098600)
Affinity DataIC50:  2.96E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by ADHP pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236981(CHEMBL4086580)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by ADHP pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236980(CHEMBL4097499)
Affinity DataIC50:  6.13E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by ADHP pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50236984(CHEMBL4069250)
Affinity DataIC50:  6.88E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by ADHP pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed