Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50049264
TargetLeucyl-cystinyl aminopeptidase(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50236826(CHEMBL4065841)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant human IRAP expressed in GnT1 deficient HEK293S cells using L-leucine 7-amido-4-methyl coumarin as substrate after 5 to 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum aminopeptidase 2(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50236826(CHEMBL4065841)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human ERAP2 using L-arginyl-7-amido-4-methyl coumarin as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2019
Entry Details Article
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50236826(CHEMBL4065841)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-leucine 7-amido-4-methyl coumarin as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2019
Entry Details Article
PubMed