Compile Data Set for Download or QSAR
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Found 22 Enz. Inhib. hit(s) with all data for entry = 50049105
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234537(CHEMBL4082042)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234540(CHEMBL4088515)
Affinity DataIC50:  20nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234538(CHEMBL4078996)
Affinity DataIC50:  39nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234552(CHEMBL4083160)
Affinity DataIC50:  40nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234549(CHEMBL4098679)
Affinity DataIC50:  40nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234544(CHEMBL4061304)
Affinity DataIC50:  40nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234557(CHEMBL4080637)
Affinity DataIC50:  50nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234558(CHEMBL4064395)
Affinity DataIC50:  50nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234551(CHEMBL4061293)
Affinity DataIC50:  50nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234543(CHEMBL4069973)
Affinity DataIC50:  60nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234546(CHEMBL4096229)
Affinity DataIC50:  70nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234554(CHEMBL4059525)
Affinity DataIC50:  70nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234547(CHEMBL4068957)
Affinity DataIC50:  70nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234556(CHEMBL4099593)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234542(CHEMBL4101403)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234541(CHEMBL4082263)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234548(CHEMBL4074097)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234545(CHEMBL4072691)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234553(CHEMBL4077380)
Affinity DataIC50:  87nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234555(CHEMBL4097016)
Affinity DataIC50:  90nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234550(CHEMBL4088508)
Affinity DataIC50:  90nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50234539(CHEMBL4064458)
Affinity DataIC50:  90nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed