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Found 16 Enz. Inhib. hit(s) with all data for entry = 50048293
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212226(CHEMBL3968176)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212224(CHEMBL3949548)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212219(CHEMBL3940787)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212227(CHEMBL3921772)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212240(CHEMBL3897016)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212223(CHEMBL3939721)
Affinity DataIC50:  4nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212225(CHEMBL3948981)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212233(CHEMBL3978113)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212230(CHEMBL3972908)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212241(CHEMBL3927260)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212220(CHEMBL3897488)
Affinity DataIC50:  7nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212221(CHEMBL3912791)
Affinity DataIC50:  12nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212242(CHEMBL3969272)
Affinity DataIC50:  15nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212228(CHEMBL3958190)
Affinity DataIC50:  20nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212222(CHEMBL3930705)
Affinity DataIC50:  24nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50212229(CHEMBL3968649)
Affinity DataIC50:  28nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential yielding 20 to 50% inactivation measured after 3 mins by patchXpress electr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed