Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50000010
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239157(CHEMBL4070666)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239157(CHEMBL4070666)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239157(CHEMBL4070666)
Affinity DataIC50: 370nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239153(CHEMBL4085518)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239158(CHEMBL4079738)
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239158(CHEMBL4079738)
Affinity DataIC50: 1.90E+4nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239156(CHEMBL4067904)
Affinity DataIC50: 2.50E+4nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239154(CHEMBL4097763)
Affinity DataIC50: 2.60E+4nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239154(CHEMBL4097763)
Affinity DataIC50: 2.60E+4nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239153(CHEMBL4085518)
Affinity DataIC50: 3.30E+4nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239154(CHEMBL4097763)
Affinity DataIC50: 4.88E+4nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239156(CHEMBL4067904)
Affinity DataIC50: 7.40E+4nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239159(CHEMBL4090048)
Affinity DataIC50: 1.02E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239155(CHEMBL4068971)
Affinity DataIC50: 1.36E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239156(CHEMBL4067904)
Affinity DataIC50: 1.52E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239159(CHEMBL4090048)
Affinity DataIC50: 1.71E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239155(CHEMBL4068971)
Affinity DataIC50: 2.57E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239155(CHEMBL4068971)
Affinity DataIC50: 3.80E+5nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239158(CHEMBL4079738)
Affinity DataIC50: 5.22E+5nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50054481((S)-2-[2-((S)-2-{(S)-2-[2-((S)-2-Amino-5-guanidino...)
Affinity DataIC50: 5.46E+5nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50054481((S)-2-[2-((S)-2-{(S)-2-[2-((S)-2-Amino-5-guanidino...)
Affinity DataIC50: 6.19E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3 (unknown origin) expressed in HEK293 cells assessed as reduction in cell adhesion to fibrinogen after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50054481((S)-2-[2-((S)-2-{(S)-2-[2-((S)-2-Amino-5-guanidino...)
Affinity DataIC50: 7.53E+5nMAssay Description:Antagonist activity at integrin alphaVbeta3alphaVbeta5 (unknown origin) expressed in SKOV3 cells assessed as reduction in cell adhesion to fibrinogen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239153(CHEMBL4085518)
Affinity DataIC50: 1.73E+6nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM50239159(CHEMBL4090048)
Affinity DataIC50: 2.95E+6nMAssay Description:Antagonist activity at integrin alphaVbeta5 (unknown origin) expressed in HT-29 cells assessed as reduction in cell adhesion to vitronectin after 2 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2019
Entry Details Article
PubMed