Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50000082
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240271(CHEMBL4101954)
Affinity DataIC50:  0.330nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240270(CHEMBL4099922)
Affinity DataIC50:  1.70nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240274(CHEMBL4092174)
Affinity DataIC50:  2nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240274(CHEMBL4092174)
Affinity DataIC50:  2.10nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM244039(10-((5-chloro-4-(2-(isopropylsulfonyl)phenyl)amino...)
Affinity DataIC50:  2.20nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM244025(9-((5-chloro-4-(2-(isopropylsulfonyl)phenyl)aminop...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM244025(9-((5-chloro-4-(2-(isopropylsulfonyl)phenyl)aminop...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM244039(10-((5-chloro-4-(2-(isopropylsulfonyl)phenyl)amino...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240276(CHEMBL4083964)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240270(CHEMBL4099922)
Affinity DataIC50:  6nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240272(CHEMBL4063965)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240271(CHEMBL4101954)
Affinity DataIC50:  11nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM244040(5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(9-me...)
Affinity DataIC50:  12nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM244040(5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(9-me...)
Affinity DataIC50:  14nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50436850(CERITINIB | CHEMBL2403108 | LDK378 | US10053458, C...)
Affinity DataIC50:  14nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240272(CHEMBL4063965)
Affinity DataIC50:  21nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240276(CHEMBL4083964)
Affinity DataIC50:  21nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50436850(CERITINIB | CHEMBL2403108 | LDK378 | US10053458, C...)
Affinity DataIC50:  24nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240273(CHEMBL4091729)
Affinity DataIC50:  29nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240273(CHEMBL4091729)
Affinity DataIC50:  130nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240269(CHEMBL4062738)
Affinity DataIC50:  190nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240275(CHEMBL4074115)
Affinity DataIC50:  260nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240269(CHEMBL4062738)
Affinity DataIC50:  300nMAssay Description:Inhibition of insulin receptor kinase (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240275(CHEMBL4074115)
Affinity DataIC50:  310nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240268(CHEMBL4100875)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type ALK (unknown origin) using TK as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50240268(CHEMBL4100875)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed